Compound ID | 2410
Class: Antimicrobial peptide
Spectrum of activity: | Gram-positive |
Details of activity: | Active against methicillin-resistant Staphylococcus epidermidis, methicillin-resistant Staphylococcus aureus, vancomycin-resistant Enterococci, Escherichia coli, Pseudomonas aeruginosa; membrane-active agent (cytoplasmic membrane) |
Description: | Synthetic compound (peptidomimetic); high selectivity towards bacterial membrane vs mammalian membrane |
Year first mentioned: | 2018 |
Development status: | Experimental |
External links: | |
Citation: | https://pubs.acs.org/doi/10.1021/acs.jmedchem.7b01704 |