Compound ID | 3574
Synonym(s): DCB-001 | DCB 001
Class: Small molecule antibacterial agent
Spectrum of activity: | Gram-positive |
Details of activity: | Active against Staphylococcus aureus including multidrug-resistant strains and methicillin-resistant strains |
Propensity to select resistant mutants: | No |
Description: | Synthetic compound; trichloroacetimidamide (TriCA2); N-(azol-2-yl)imidamide scaffold; shows efficacy in treating methicillin-resistant Staphylococcus aureus bacteraemia infection model with comparable outcomes to vancomycin and ampicillin |
Institute where first reported: | DimiCare Biotech (Nice, France) |
Development status: | Experimental |
External links: | |
Citation: | https://www.dimicare-biotech.com/pipeline/ |